经验分子式(希尔表示法) C27H45IN2
分子量 524.56
MDL number MFCD07370143
IC50 = 60 nM for eEF-2 kinase vs protein kinase C (IC50= 7.5 μM), protein kinase A (IC50= 80 μM), and calmodulin-dependent kinase II IC50 > 100 μM).
NH125 is a novel plant histidine kinase inhibitor and selective mammalian eurkaryotic elongation factor-2 kinase (eEF-2K).
在氮气保护下封装。
assay | ≥98% (HPLC) |
form | solid |
color | white to off-white |
mp | 88.2-94.9 °C |
solubility | DMSO: >20 mg/mL |
storage temp. | ?20°C |
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