经验分子式(希尔表示法) C27H32N6O
分子量 456.58
CINK4 is a specific inhbitor of CDK4/cyclin D1 complexes (IC50 = 1.5 mM). CINK4 has greater than 50 fold selectivity over CDK1 or CDK2. CINK4 dose-dependently inhibits phosphorylation of retinoblastoma (Rb) and induces G0-G1 cell cycle arrest and apoptosis in cancer cell lines.
assay | ≥95% (HPLC) |
form | powder |
color | white to light brown |
solubility | DMSO: soluble25 mg/mL, clear |
storage temp. | 2-8°C |
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