经验分子式(希尔表示法) C14H21N5O2S
分子量 323.41
This compound was developed by Pfizer for Kinase Phosphatase Biology research. To learn more about Sigma′s partnership with Pfizer and view other authentic, high-quality Pfizer compounds, visit sigma.com/bsm-pfizer.
Sold for research purposes under agreement from Pfizer Inc.
PF-04965842 is a Janus Kinase (JAK) inhibitor selective for JAK1 with an IC50 value of 29 nM for JAK1 compared to 803 nM for JAK2, >10000 nM for JAK3 and 1250 nM for Tyk2. JAKs mediate cytokine signaling, and are involved in cell proliferation and differentiation. PF-04965842 has been investigated as a possible treatment for psoriasis.
assay | ≥98% (HPLC) |
form | powder |
color | white to beige |
solubility | DMSO: soluble10 mg/mL, clear |
storage temp. | room temp |
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