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产品名称
omega-Agatoxin TK,Ca V2.1 P/Q-type calcium channel blocker
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描述
Potent,selective Ca V2.1 P/Q-type calcium channel blocker
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生物学描述
Potent, selective Ca V2.1 P/Q-type calcium channel blocker (Kd = 3 nM, P-type). Inhibits the high K + depolarisation-induced rise in internal Ca 2+ in nerve endings (IC 50 = 60 nM) .
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纯度
> 99%
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CAS编号
158484-42-5
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化学结构