属于速激肽家族的神经介素L是比P物质更有效的支气管收缩剂,并可调节中性粒细胞募集到下呼吸道。
序列(三个字母) | H-Gly-Tyr-Pro-Gly-Gln-Val-OH |
序列(一个字母) | GYPGQV |
CAS | [225779-44-2] |
纯度 | ≥95.0% |
分子量 | 619.7 |
Description | This peptide is the amino terminus of the fourth protease-activated receptor (PAR4) after the cleavage at Arg47/Gly48 was tested for its ability to stimulate COS cells expressing PAR4. The peptide readily activated both wild-type and mutant PAR4 (R47A) at 500 ?M, whereas thrombin and trypsin only activate the wild-type PAR4. |
Formula | C28H41N7O9 |
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