0
| Replacement Information |
|---|
| Empirical Formula | CAS # |
|---|---|
| C₁₈H₁₄BrN₅O₆PS · Na | 172806-20-1 |
| Description | |
|---|---|
| Overview | A metabolically-stable, competitive inhibitor of protein kinase G types 1α and 1β (Ki = 30 nM). Blocks cGMP-gated retinal type ion channels (IC50 = 25 µM) and the activation of purified PKA type II (Ki = 10 µM). More lipophilic and cell-permeable than Rp-8-pCPT-cGMPS (Cat. No. 370677). Note: 1 µmol = 0.56 mg. |
| Catalogue Number | 370679 |
| Brand Family | Calbiochem® |
| Synonyms | Rp-8-Br-PET-cGMPS, Na, PKG Inhibitor VI |
| References | |
|---|---|
| References | Wei, J.Y., et al. 1996. Biochemistry 35, 16815. Butt, E., et al. 1995. Br. J. Pharmacol. 116, 3110. |
| Applications |
|---|
| Biological Information | |
|---|---|
| Primary Target | PKG1α & 1β |
| Primary Target K<sub>i</sub> | 30 nM against PKG1α & 1β |
| Purity | ≥98% by HPLC |
| Physicochemical Information | |
|---|---|
| Cell permeable | Y |
| Dimensions |
|---|
| Materials Information |
|---|
| Toxicological Information |
|---|
| Safety Information according to GHS |
|---|
| Safety Information |
|---|
| Product Usage Statements |
|---|
| Packaging Information |
|---|
| Transport Information |
|---|
| Supplemental Information |
|---|
| Specifications |
|---|
温馨提示:因厂家更改产品包装、产地或者更换随机附件等没有任何提前通知，且每位咨询者购买情况、提问时间等不同，为此以下回复仅对提问者3天内有效，其他网友仅供参考！若由此给您带来不便请多多谅解，谢谢！
服务热线
0771-3293894
新浪微博
腾讯微博
QQ空间
客服
