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Qiagen 凯杰 Biosharp Omega

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Membrane Transporter/Ion Channel Compound Library 50μL/well(10mM solution)

价:
0.00
价:
¥0.00

号:HY-L011

牌:MCE

账期 货到付款

(预计4-5工作日到货(以MCE官网货期为准))

亲,想了解价格请QQ咨询客服!

工作时间

周一至周五:9:00-18:00

咨询电话

0771-3293894

在线咨询

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Description
& Advantages

•   A unique collection of 416 small molecule modulators used for Ion Channel and Membrane Transporter research.

•   The library contains compounds targeting Membrane Transporters including Pgp, CRM1, BCRP, etc., and Ion Channels including CFTR, proton pump, sodium pump, calcium pump, etc.

•   A useful tool for the research of drug absorption and distribution.

•   Bioactivity and safety confirmed by preclinical research and clinical trials. Some inhibitors have been approved by FDA.

•   Structurally diverse, medicinally active, and cell permeable.

•   Rich documentation with structure, IC50, and summary.

•   NMR and HPLC validated to ensure high purity.

•   All compounds are in stock and continuously updated.

Product Details
Formulation:
A collection of 416 Membrane Transporter/Ion Channel related compounds supplied as pre-dissolved DMSO solutions or Solid
Container:
96 Well Format Sample Storage Tube With Screw Cap and Optional 2D Barcode
Storage:
-80°C
Shipping:
Blue ice
Composition

Membrane Transporter/Ion Channel Compound Library

Source: MedChem Express

Contents of Membrane Transporter/Ion Channel Compound Library

Plate layout: HY-L011-1

1 2 3 4 5 6 7 8 9 10 11 12
a Empty SKF-96365 (hydrochloride) Vonoprazan Ko 143 JNJ-17203212 Pipequaline PAP-1 HC-067047 SKF89976A (hydrochloride) DMCM (hydrochloride) MRK-016 Empty
b Empty LY2365109 (hydrochloride) ZL006 A-804598 CaCCinh-A01 U93631 D-AP5 GSK2193874 Norverapamil (hydrochloride) gamma-DGG Kynurenic acid Empty
c Empty Isoguvacine (hydrochloride) 7-Chloro-4-hydroxyquinoline-2-carboxylic acid 7-Chlorokynurenic acid sodium salt YM-58483 Diphenyleneiodonium chloride NPPB Sarcosine Allopregnanolone Sodium ionophore III Org-26576 Empty
d Empty DHBP (dibromide) ZD7288 PF-01247324 Picrotoxin ICA-069673 4-Acetamidobutanoic acid L-DABA Vanilpyruvic acid GAL-021 Bamaquimast Empty
e Empty NS-638 CDN1163 Polyoxyethylene stearate Ilaprazole AMG9810 EIPA ML213 PSB-12062 GYKI53655 hydrochloride Bepridil hydrochloride Empty
f Empty CGP52432 Gabazine ML335 Capsaicin Dapagliflozin Dapagliflozin ((2S)-1,2-propanediol, hydrate) Canagliflozin Fantofarone Tariquidar Tariquidar (methanesulfonate, hydrate) Empty
g Empty Ketanserin Ketanserin (tartrate) Eniporide hydrochloride SB-705498 AMG 517 Almitrine mesylate Kynurenic acid (sodium) SN 6 Desformylflustrabromine hydrochloride Aminooxyacetic acid hemihydrochloride Empty
h Empty Mirogabalin besylate Bitopertin AM-0902 WS-12 A-967079 Pyr3 Aniracetam LY450108 Farampator NS11394 Empty

Plate layout: HY-L011-2

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Icilin A-803467 A-867744 NS 1738 PNU-120596 ABT-239 SB-366791 Rostafuroxin PEAQX (tetrasodium hydrate) ML277 Empty
b Empty NS-1619 (S)-Willardiine Efonidipine (hydrochloride monoethanolate) CFM-2 Pyr6 CX546 Naspm Naspm (trihydrochloride) GSK-7975A PEPA Empty
c Empty Nicardipine (Hydrochloride) Dantrolene (sodium hemiheptahydrate) PNU-282987 GS967 Hexachlorophene R(+)-IAA-94 LDN-212320 AZD3965 YHO-13177 YHO-13351 (free base) Empty
d Empty Optovin Eliprodil Ifenprodil (tartrate) ML204 ML204 (hydrochloride) Ivacaftor SDZ 220-581 SDZ 220-581 (hydrochloride) RJR-2403 (hemioxalate) VX-809 Empty
e Empty KN-62 Vinpocetine Tofogliflozin (hydrate) Zatebradine (hydrochloride) Zatebradine TRAM-34 Cisatracurium (besylate) HM30181 Lansoprazole (R)-Lansoprazole Empty
f Empty MRX-1024 A 839977 Ro 25-6981 (Maleate) PPQ-102 Amiodarone (hydrochloride) Levcromakalim Nilvadipine Pinacidil monohydrate Tebanicline (hydrochloride) L-655708 Empty
g Empty Sibutramine (hydrochloride) AF-353 GTS-21 (dihydrochloride) Rosiglitazone (maleate) Diltiazem (hydrochloride) PTC124 Phenylpiracetam Ipragliflozin AWD 131-138 HC-030031 Empty
h Empty Chembridge-5861528 CNQX DNQX NBQX ZK200775 ZK200775 (hydrate) Talampanel (+)-MK 801 (Maleate) (-)-MK 801 (Maleate) Bay-K-8644 ((S)-(-)-) Empty

Plate layout: HY-L011-3

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Bay-K-8644 ((R)-(+)-) Glibenclamide Zosuquidar Lesinurad Lesinurad (sodium) TAK-438 Vigabatrin Empagliflozin KB-R7943 (mesylate) NS309 Empty
b Empty VX-661 PF-04971729 GW791343 (dihydrochloride) UK-5099 A 438079 A 438079 (hydrochloride) LX-4211 S0859 E-4031 Mibefradil (dihydrochloride) Empty
c Empty A-317491 A-317491 (sodium salt hydrate) Capsazepine QNZ46 NS6180 CGP37157 BTB06584 Gabapentin enacarbil MDL-29951 Transcrocetinate disodium Empty
d Empty Etifoxine (hydrochloride) Etifoxine CFTR(inh)-172 VU 0240551 SN 2 (S)-(-)-5-Fluorowillardiine (hydrochloride) Verinurad ICA-121431 NS1643 Flupirtine (Maleate) Empty
e Empty Dofequidar (fumarate) Acamprosate (calcium) (R)-Baclofen Valspodar Rosiglitazone Mitiglinide (Calcium) Ranolazine (dihydrochloride) Manidipine (dihydrochloride) Cilnidipine Vinblastine Empty
f Empty Flecainide (acetate) Clevidipine Noopept Bumetanide Pantoprazole (sodium) Sunifiram NMDA Coluracetam Meclofenoxate (hydrochloride) Nonivamide Empty
g Empty Radafaxine (hydrochloride) Bexagliflozin GlyH-101 IOWH-032 Azimilide (Dihydrochloride) RQ-00203078 SYM2206 L-701324 CIQ GlyT2-IN-1 Empty
h Empty Adjudin Lorediplon Pyr10 GSK1016790A Cariporide KS176 XEN907 BCTC KM11060 RN-1734 Empty

Plate layout: HY-L011-4

1 2 3 4 5 6 7 8 9 10 11 12
a Empty CRAC intermediate 2 (-)-Aspartic acid Transcrocetin meglumine salt Zosuquidar (trihydrochloride) Senicapoc A-740003 Elacridar Proparacaine (Hydrochloride) Dronedarone (Hydrochloride) Gabapentin Empty
b Empty Gabapentin (hydrochloride) Verapamil (hydrochloride) Tetracaine Trimethadione Mexiletine (hydrochloride) Flumazenil Azelnidipine Vigabatrin (Hydrochloride) Etomidate Etomidate (hydrochloride) Empty
c Empty Levetiracetam Minoxidil Omeprazole Oxcarbazepine Vecuronium (bromide) Zonisamide Furosemide Prilocaine Felbamate Lidocaine Empty

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