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Qiagen 凯杰 Biosharp Omega

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GPCR/G Protein Compound Library 30μL/well(10mM solution)

价:
0.00
价:
¥0.00

号:HY-L006

牌:MCE

账期 货到付款

(预计4-5工作日到货(以MCE官网货期为准))

亲,想了解价格请QQ咨询客服!

工作时间

周一至周五:9:00-18:00

咨询电话

0771-3293894

在线咨询

客服 郭恒 蔡玉坤 曾宪飞 技术咨询

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Description
& Advantages

•   A unique collection of 728 small molecules targeting G protein coupled receptors used in GPCR screening for various research and drug development projects.

•   Targets such as 5-HT Receptor, Dopamine Receptor, Opioid Receptor, Adrenergic Receptors, Cannabinoid Receptor, mGluR, ETA Receptor, etc.

•   The most successful class of drugable targets in the human genome and remain the most attractive family of targets.

•   All of the small molecules in the GPCR library are well characterized with biological and pharmaceutical activity. Some compounds have been approved by the FDA.

•   A powerful tool for discovering GPCR-based drugs that are the richest signal receptor targets for drug discovery.

•   Structurally diverse, medicinally active, and cell permeable.

•   Rich documentation with structure, IC50, and brief introduction.

•   NMR and HPLC validated to ensure the highest purity.

•   All compounds are in stock and continuously updated.

Product Details
Formulation:
A collection of 728 GPCR/G Protein related compounds supplied as pre-dissolved DMSO solutions or Solid
Container:
96 Well Format Sample Storage Tube With Screw Cap and Optional 2D Barcode
Storage:
-80°C
Shipping:
Blue ice
Composition

GPCR/G Protein Compound Library

Source: MedChem Express

Contents of GPCR/G Protein Compound Library

Plate layout: HY-L006-1

1 2 3 4 5 6 7 8 9 10 11 12
a Empty PD 117519 NPS-2143 Taranabant 4-IBP DREADD agonist 21 Lu AF21934 (RS)-MCPG SQ22536 Ro 67-7476 (S)-MCPG Empty
b Empty JNJ16259685 PHCCC TCS-OX2-29 Plerixafor Bay 59-3074 Aprepitant Flopropione VU0364770 Ticagrelor YL0919 Empty
c Empty Piperoxan (hydrochloride) Zibotentan ONO-7300243 Norbinaltorphimine dihydrochloride ZK756326 (dihydrochloride) AR-M 1000390 (hydrochloride) Ocaperidone SB-224289 hydrochloride Naltrindole (hydrochloride) Vorapaxar Empty
d Empty GSK682753A Silodosin Agmatine (sulfate) ST034307 Phenylbiguanide Ro 10-5824 (dihydrochloride) Nicotinamide N-oxide Vanilpyruvic acid CYM-5541 VUF10460 Empty
e Empty IT1t (dihydrochloride) GPR120-IN-1 NPS-2143 (hydrochloride) Veralipride N6-(2-Phenylethyl)adenosine BQCA CB-7921220 AVex-73 hydrochloride DC260126 Prostaglandin E2 Empty
f Empty Navarixin AZD4635 (RS)-Butyryltimolol PD 123319 (ditrifluoroacetate) TC-G-1008 MK-3207 (Hydrochloride) E7046 SB-399885 hydrochloride LY334370 NECA Empty
g Empty SB297006 WAY-100635 Maleate BETP 1A-116 MK-2894 MK-2894 (sodium salt) AH 6809 SKF-82958 (hydrobromide) TAK-875 JDTic (dihydrochloride) Empty
h Empty DADLE Ketanserin Ketanserin (tartrate) Sarpogrelate (hydrochloride) Ponesimod Palosuran MK-6892 Pridopidine Asimadoline VU 0365114 Empty

Plate layout: HY-L006-2

1 2 3 4 5 6 7 8 9 10 11 12
a Empty CGP71683 hydrochloride Methiothepin mesylate CJ-42794 Almorexant Almorexant (hydrochloride) Teijin compound 1 (Z)-Thiothixene CCG-203971 Otenabant Istradefylline Empty
b Empty Preladenant RO1138452 SB-334867 (free base) SB-674042 TCS 1102 Tozadenant Fingolimod Asenapine (maleate) Sitaxsentan (sodium) ONC212 Empty
c Empty ALB-127158(a) LP-211 Desisobutyryl-ciclesonide 8-OH-DPAT Chlorcyclizine (hydrochloride) N-Acetylhistamine VU0467154 AZ3451 Fingolimod (hydrochloride) 3-Isopropyl-5-(4-(((6-(4-(methylsulfonyl)phenyl)pyridin-3-yl)oxy)methyl)piperidin-1-yl)-1,2,4-oxadiazole Empty
d Empty BX471 VU 0238429 JNJ-5207852 ABT-239 Pitolisant (hydrochloride) Ozanimod MK-3697 Siponimod 2-Cl-IB-MECA BAY 41-2272 Empty
e Empty Atipamezole (hydrochloride) Atipamezole Angiotensin (1-7) 6H05 (trifluoroacetate) SKF 38393 (hydrochloride) Terlipressin Gonadorelin (acetate) Y16 Prucalopride (succinate) Bromocriptine (mesylate) Empty
f Empty Piribedil Rauwolscine (hydrochloride) Trimethobenzamide hydrochloride ML141 EHop-016 RBC8 CASIN BQU57 Dinoprost (tromethamine salt) Batefenterol Empty
g Empty Pimozide MK-0354 SRT3190 ADL-5859 ADX-47273 (R)-ADX-47273 MRS 2578 WAY-100635 (maleate salt) CGS 21680 (Hydrochloride) Biperiden (Hydrochloride) Empty
h Empty MTEP (hydrochloride) Ambrisentan AM211 BRL 54443 BAN ORL 24 PF-4136309 JTC-801 Ki16425 Org 27569 WIN 55,212-2 (Mesylate) Empty

Plate layout: HY-L006-3

1 2 3 4 5 6 7 8 9 10 11 12
a Empty Montelukast (sodium) VU0152100 TAK-779 SB 242084 SB 242084 (hydrochloride) Xanomeline (oxalate) SR144528 PF429242 (dihydrochloride) Nedocromil JNJ-7777120 Empty
b Empty SA4503 (dihydrochloride) Rupatadine (Fumarate) LY310762 Abarelix Betamethasone Betamethasone dipropionate Beclometasone dipropionate Budesonide Clobetasol propionate Deflazacort Empty
c Empty Leuprolide Acetate Goserelin (acetate) Mifepristone Mometasone furoate MSX-122 Norepinephrine (bitartrate monohydrate) Noscapine Pergolide (mesylate) LY 344864 LY 344864 racemate Empty
d Empty IPSU BPTU Angiotensin II human ICI 118,551 (hydrochloride) Telmisartan ZCL278 AMG 837 (calcium hydrate) UNC0642 CCG-1423 CP 376395 Empty
e Empty Rimonabant (Hydrochloride) Aclidinium (Bromide) Cisapride Prucalopride Tegaserod (maleate) GW842166X Macitentan Lixivaptan TGR5 Receptor Agonist Vilazodone (Hydrochloride) Empty
f Empty Vilazodone Lodoxamide Indacaterol (maleate) Salmeterol SB 271046 (Hydrochloride) SB-742457 AC-55541 Elagolix sodium (1R,2S)-VU0155041 VU0361737 Empty
g Empty TCN238 MLE-4901 Bilastine JNJ-31020028 Latrepirdine (dihydrochloride) Haloperidol Clozapine Olanzapine Sertindole Quetiapine Empty
h Empty Amisulpride Aripiprazole Talnetant Pimavanserin Pimavanserin tartrate Tandospirone TBPB L-Glutamic acid monosodium salt MPEP (Hydrochloride) CPPHA Empty

Plate layout: HY-L006-4

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1 2 3 4 5 6 7 8 9 10 11 12
a Empty Dexamethasone Dexamethasone (acetate) Anamorelin Anamorelin (hydrochloride) Rolapitant Salirasib Cariprazine Cariprazine (hydrochloride) Mirabegron Riociguat Empty
b Empty Adoprazine Elagolix (±)-SLV319 Tasimelteon Tarafenacin (D-tartrate) Lasmiditan (hydrochloride) NS-304 Taprenepag Azilsartan Lificiguat Empty
c Empty Volinanserin OPC-21268 PF-3274167 Sinomenine hydrochloride O-Phospho-L-serine